Ite elegbogi ti o ga julọ 1421373-66-1 Mesylate-AZD9291 fun Itọju Akàn
Ọjaoruko | AZD-9291 mesylate |
Awọn itumọ ọrọ sisọ | N-[2-[[2- (Dimethylamino) ethyl] methylamino] -4-methoxy-5-[[4- (1-methyl-1H-indol-3-yl) -2-pyrimidinyl] amino] phenyl] - 2-propenamide methanesulfonate (1:1) |
CAS No. | 1421373-66-1 |
Ifarahan | Funfun si ina ofeefee ri to lulú |
Fọọmu Molecular | C28H33N7O2.CH4O3S |
Òṣuwọn Molikula | 595.71 |
Lilo | Elegbogi ite tabi Iwadi idi |
Iṣakojọpọ | Gẹgẹbi ibeere rẹ |
Ibi ipamọ | Fipamọ ni wiwọ, awọn apoti sooro ina ni aye tutu |
AZD-9291 mesylateCAS: 1421373-66-1 | ||
Items | Standards | Rawọn abajade |
Ifarahan | Funfun si ina ofeefee ri to lulú | Ina ofeefee ri to lulú |
Ieyin | Nipasẹ IR | Ibamu |
Nipasẹ HPLC | Ibamu | |
Solubility | Soluble ni Dimethylsulfoxide, tiotuka die-die ni Ethanol ati Acetonitrile, pẹlu pH ti o gbẹkẹle solubility olomi | Ibamu |
Akoonu Omi(KF) | ≤ 1.00% | 0.42% |
Aloku lori Iginisonu | ≤ 0.10% | 0.05% |
HrọrunMetal | 20ppm | Ibamu |
Mesylate | 15.20% ~ 18.20% | 15.90% |
Awọn ohun elo ti o ku | Acetonitrile: ≤410ppm | ND |
Acetone: ≤5000ppm | ND | |
Tetrahydrofuran: ≤720ppm | ND | |
Rinu didunSohun elo | O pọju ẹyọkan alaimọ: ≤0.20% | 0.17% |
Lapapọ awọn idoti: ≤1.00% | 0.25% | |
Patiku Iwon | D90: ≤100μm | 57.97% |
Asọ (HPLC ipilẹ lori gbigbe) | 98.00% ~ 102.00% | 99.80% |
Standard itọkasi | Ni-ile Standard |
Ile-iṣẹ Alaye
√ Iriri kikun ti Layer iṣakoso ni ile-iṣẹ ati awọn ọmọlẹyin awọn onimọ-ẹrọ oye; √ Didara nigbagbogbo jẹ akiyesi oke wa, Eto QC to muna; √ 11 ọdun ti o ni iriri ẹgbẹ tita ọja okeere; √ Lab R&D olominira; √ Awọn idanileko GMP igba pipẹ ti a fowo si; √ Awọn orisun ọlọrọ ti ọpọlọpọ awọn ile-iṣelọpọ laišišẹ fun iṣẹ akanṣe; √ Ẹgbẹ iṣẹ ṣiṣe ti o ga julọ pẹlu ọna deede.Kọ ifiranṣẹ rẹ nibi ki o si fi si wa